OtherPeptideEvidence C2 cited

AHK-Cu

Alanine-Histidine-Lysine Copper Peptide

aka Copper tripeptide AHK · Ala-His-Lys-Cu

A synthetic copper tripeptide analogue of GHK-Cu, researched for collagen synthesis and skin regeneration.

Molecular wt
451.39g/mol
Formula
C15H24ClCuN6O4-
CAS
682809-81-0
Route
Topical / subcutaneous

Sequence

One-letter3 residues

AHK

Three-letter

L-Ala-L-His-L-Lys

Read this before quoting the sequence
Tripeptide L-alanyl-L-histidyl-L-lysine complexed with copper(II). The free tripeptide AHK is PubChem CID 7408502 (C15H26N6O4, 354.41 g/mol). The copper complex is a coordination compound, not a plain peptide, and its stoichiometry/counter-ion vary between preparations.
Source ↗

Mechanism of action

AHK-Cu is a copper tripeptide that binds to copper ions, facilitating their transport into cells. This peptide enhances the activity of enzymes involved in collagen synthesis and tissue repair. It also modulates the expression of genes related to skin regeneration and anti-inflammatory responses. AHK-Cu is more stable than its parent compound, GHK-Cu, allowing for prolonged activity in biological systems.

What the evidence actually shows

Grade C

There are no human clinical trials specifically evaluating AHK-Cu. Most evidence comes from in vitro studies and animal models demonstrating its effects on skin and hair. The lack of human data limits the ability to fully understand its efficacy and safety profile.

Regulatory status

Status
Not an approved drug in any jurisdiction identified. Used as a cosmetic ingredient; no registered human clinical trial found on ClinicalTrials.gov.
Clinical stage
Preclinical / in vitro and ex vivo only
UK
research_compound

AHK-Cu is not approved by the MHRA for medical use and is considered a research compound.

Source ↗

Dosing — what backs each figure

AHK-Cu has no human dosing of any kind. The single substantive study exposed cultured human dermal papilla cells and ex-vivo hair follicles to 1e-12 to 1e-9 M peptide in the culture dish — a concentration, not a dose. Nothing supports administering it by injection, and no clinical trial has been run.

PreclinicalAnimal studies — not a human dose
  • 1e-12 M to 1e-9 M in culture medium; stimulated elongation of human hair follicles ex vivo and proliferation of dermal papilla cells in vitro

    human tissue ex vivo / human dermal papilla cells in vitro (not a live-organism dose) · added to culture medium · PMID 17703734

Animal doses do not convert to human doses by body weight alone. Route matters too — a compound dosed intraperitoneally in mice tells you little about subcutaneous use.

Commonly circulatedNot established by any study
Dose
1-3 mg/day (topical); 100-500 mcg/day (SubQ)
Frequency
Daily
Cycle
8-12 weeks· unsourced

Why this isn't evidence
AHK-Cu is a topical cosmetic ingredient whose only published data are picomolar-to-nanomolar concentrations in cell and ex-vivo follicle culture; there is no in-vivo dose in ANY species, so both the mg/day topical figure and the subcutaneous mcg/day figure are unsourced, and quoting an injectable dose for a cosmetic ingredient is a category error.

This figure is shown because it is what circulates and what people search for — not because it is supported. Cycle lengths in particular tend to be convention copied between compounds rather than anything derived from a compound's own pharmacokinetics.

No established human dose
No approved label or completed human trial establishes a dosing regimen for this compound. Anything presented as a standard protocol for it — anywhere — is someone's convention rather than a finding.

Handling and storage

No compound-specific stability data exists
No stability/storage study for AHK-Cu was located in a primary or regulatory source. No compound-specific stability study (lyophilised or reconstituted) was located in a primary/regulatory source during this verification pass. Only generic synthetic-peptide handling guidance exists for this compound; no specific temperatures or durations are recorded here rather than fabricating them. General peptide handling still applies — reconstitute gently, keep it cold, keep it dark — but any specific figure you see quoted for this compound elsewhere is someone's assumption, not a measurement.

Safety

Commonly reported
  • ·Mild skin irritation
Rarely reported
  • ·Allergic reactions
Contraindications
  • ·Known hypersensitivity to copper peptides
Drug interactions
  • ·Chelating agents may reduce effectiveness by binding copper ions

Reported combinations

Reported as synergistic
  • ·Vitamin C, which supports collagen synthesis
Reported as antagonistic
  • ·Chelating agents

Combination claims in this dataset are largely unsourced and should be treated as folk knowledge until a citation appears beside them.

References (2)

Data provenance

Chemistry and citations on this page were checked against primary sources on 2026-08-14. Values that could not be verified were left blank rather than filled with a plausible guess.

Could not verify
storage.lyophilized, storage.reconstituted, storage.lightSensitive, reconstitution.solvent, regulatory.wada

Research use only
This profile is educational reference material. It is not medical advice, not a prescription, and not an endorsement of self-administration. Compounds discussed here are research chemicals and most are not approved for human therapeutic use.